The invention discloses a dialkyl and diaryl tetrasubstituted
heterocyclic compound, their preparing process and use, the compound has the general formula disclosed in the specification, wherein X is selected from S, O, NH and N-
alkyl derivative, R1, R5, R'1, R'4, R'5 are selected from H, R6, R'5 are selected from
alkyl, in particular
alkyl of C1-C4, R2 is selected from H, methoxyl, R3 is selected from
halogen, alkoxy, in particular alkyl of C1-C4 and PhCH2-alkoxy, R4 is selected from H, methoxyl,
halogen, R'2 is selected from H, methoxyl,
halogen and amine derivative, R'3 is selected from halogen, alkoxy, in particular alkyl of C1-C4 and PhCH2-alkoxy. The substituted
heterocyclic compound can be used in preparing medicinal compositions, especially medicament for antineoplastic and anti-inflammatory actions.